2. Signaling Pathways
  3. GPCR/G Protein
    Neuronal Signaling
  4. Melanocortin Receptor
  5. MC2R Isoform
  6. MC2R Antagonist

MC2R Antagonist

MC2R Antagonist (1):

Cat. No. Product Name Effect Purity
  • HY-158081
    CRN04894
    		Antagonist 98.41%
    CRN04894 (compound 17h) is an orally active MC2R antagonist that demonstrates in vivo efficacy in rat model of adrenocorticotropic hormone (ACTH)-stimulated corticosterone secretion[1]. CRN04894 binds to human or rat MC2R with KB values of 0.34 nM and 0.23 nM, respsectively.